A1AR antagonist 6
CAT:
804-HY-147545
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
A1AR antagonist 6
- CAS Number: 329693-22-3
- UNSPSC Description: A1AR antagonist 6 (compound 15) is a potent and selective A1AR (A1 adenosine receptor) antagonist, with a pIC50 of 6.38 and a pKi of 7.13[1].
- Target Antigen: Adenosine Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein
- Applications: Neuroscience-Neuromodulation
- Field of Research: Neurological Disease
- Assay Protocol: https://www.medchemexpress.com/a1ar-antagonist-6.html
- Solubility: 10 mM in DMSO
- Smiles: N#CC1=C(N=C2CCCCC2=C1C3=CC=C4OCOC4=C3)N
- Molecular Weight: 293.32
- References & Citations: [1]Wei Y, et al. Identification of new potent A1 adenosine receptor antagonists using a multistage virtual screening approach. Eur J Med Chem. 2020 Feb 1;187:111936.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported