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SORT-PGRN interaction inhibitor 3

CAT:
804-HY-153688
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  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
SORT-PGRN interaction inhibitor 3 - image 1

SORT-PGRN interaction inhibitor 3

  • CAS Number: 2691846-87-2
  • UNSPSC Description: SORT-PGRN interaction inhibitor 3 (Compound 13) is a SORT-PGRN interaction inhibitor (IC50: 0.17 μM). SORT-PGRN interaction inhibitor 3 can be used for research of neurodegenerative diseases[1].
  • Target Antigen: Neurotensin Receptor
  • Type: Reference compound
  • Related Pathways: GPCR/G Protein;Neuronal Signaling
  • Applications: Neuroscience-Neurodegeneration
  • Field of Research: Neurological Disease
  • Assay Protocol: https://www.medchemexpress.com/sort-pgrn-interaction-inhibitor-3.html
  • Solubility: 10 mM in DMSO
  • Smiles: CC(C)(C)CC[C@@H](C(O)=O)NC(C1=CC(Cl)=CC(Cl)=C1)=O
  • Molecular Weight: 332.22
  • References & Citations: [1]Stachel SJ, et al. Identification of potent inhibitors of the sortilin-progranulin interaction. Bioorg Med Chem Lett. 2020 Sep 1;30(17):127403.
  • Shipping Conditions: Room temperature
  • Clinical Information: No Development Reported