PI3K/VEGFR2-IN-1
CAT:
804-HY-151635
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

PI3K/VEGFR2-IN-1
- CAS Number: 2851067-08-6
- UNSPSC Description: PI3K/VEGFR2-IN-1 is a potent dual PI3K/VEGFR2 inhibitor with IC50 values of 2.21 and 68 μM for PI3K and VEGFR2, respectively. PI3K/VEGFR2-IN-1 induces apoptosis. PI3K/VEGFR2-IN-1 can be used in research of cancer[1].
- Target Antigen: Apoptosis; PI3K; VEGFR
- Type: Reference compound
- Related Pathways: Apoptosis;PI3K/Akt/mTOR;Protein Tyrosine Kinase/RTK
- Applications: Cancer-Kinase/protease
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/pi3k-vegfr2-in-1.html
- Solubility: 10 mM in DMSO
- Smiles: S=C(N/N=C(C1=CC2=CC=CC=C2O1)\C)NC3=CC=C(Cl)C=C3
- Molecular Weight: 343.83
- References & Citations: [1]El-Khouly OA, et, al. Design, synthesis and computational study of new benzofuran hybrids as dual PI3K/VEGFR2 inhibitors targeting cancer. Sci Rep. 2022 Oct 12;12(1):17104.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported