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LSD1-IN-16

CAT:
804-HY-144757
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  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
LSD1-IN-16 - image 1

LSD1-IN-16

  • UNSPSC Description: LSD1-IN-16 (compound 4b) is a potent LSD1 inhibitor. LSD1-IN-16 can inhibit LSD1-CoREST, MAO-A and MAO-B, with IC50 values of 0.015, 0.024, and 0.366 μM, respectively. LSD1-IN-16 displays cell growth arrest in prostate cancer LNCaP cells, with an IC50 of 15.2 μM[1].
  • Target Antigen: Histone Demethylase; Monoamine Oxidase
  • Type: Reference compound
  • Related Pathways: Epigenetics;Neuronal Signaling
  • Applications: Cancer-programmed cell death
  • Field of Research: Cancer
  • Assay Protocol: https://www.medchemexpress.com/lsd1-in-16.html
  • Solubility: 10 mM in DMSO
  • Smiles: NC1CC1C2=CC=C(C=C2)NC(C3=CC=CC(C4=CC=CS4)=C3)=O
  • Molecular Weight: 334.43
  • References & Citations: [1]Fioravanti R, et al. Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity. J Enzyme Inhib Med Chem. 2022 Dec;37(1):973-985.
  • Shipping Conditions: Room temperature
  • Clinical Information: No Development Reported