MCT-IN-1

• CAS Number:

  1685273-57-7

• UNSPSC Description:

  MCT-IN-1 (compound 2) is a potent inhibitor of monocarboxylate transporter (MCT), with the IC50 of 9 nM and 14 nM for MCT1 and MCT4, respectively[1].

• Target Antigen:

  Monocarboxylate Transporter

• Type:

  Reference compound

• Related Pathways:

  Membrane Transporter/Ion Channel

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/mct-in-1.html

• Solubility:

  DMSO : 200 mg/mL (ultrasonic)

• Smiles:

  CCCCN(C1=CC(OC)=C(C=C1)/C=C(C#N)/C(O)=O)CCCC

• Molecular Weight:

  330.42

• References & Citations:

  [1]Sachin Puri, et al. Monocarboxylate transporter 1 and 4 inhibitors as potential therapeutics for treating solid tumours: A review with structure-activity relationship insights. Eur J Med Chem. 2020 Aug 1:199:112393.

• Shipping Conditions:

  Room Temperature

• Clinical Information:

  No Development Reported