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WDR5-IN-8

CAT:
804-HY-161123
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  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
WDR5-IN-8 - image 1

WDR5-IN-8

  • UNSPSC Description: WDR5-IN-8 is a WDR5 inhibitor with IC50 value of 15.5 nM. WDR5-IN-8 shows good anti-proliferative activity in two human acute leukemia cell lines. WDR5-IN-8 has antitumor activity[1].
  • Target Antigen: WDR5
  • Type: Reference compound
  • Related Pathways: Epigenetics
  • Applications: Cancer-programmed cell death
  • Field of Research: Cancer
  • Assay Protocol: https://www.medchemexpress.com/wdr5-in-8.html
  • Solubility: 10 mM in DMSO
  • Smiles: CC1=C(C2=C(C3=CC(NCC4=C(NC=N4)C)=C2)CCN(C3=O)CC5=CC=C(C=C5)Cl)C=C(CO)C=C1
  • Molecular Weight: 501.02
  • References & Citations: [1]Qin S, et al. Discovery and Optimization of WDR5 Inhibitors via Cascade Deoxyribonucleic Acid-Encoded Library Selection Approach. J Med Chem. 2024 Jan 3.
  • Shipping Conditions: Room temperature
  • Clinical Information: No Development Reported