CARM1-IN-6

• CAS Number:

  1269199-96-3

• UNSPSC Description:

  CARM1-IN-6 (iCARM1) is an effective and selective inhibitor of CARM1 with an IC50 value of 12.3 μM. CARM1-IN-6 exhibits cell growth inhibitory activity and can be used in cancer research[1].

• Target Antigen:

  Histone Methyltransferase

• Type:

  Reference compound

• Related Pathways:

  Epigenetics

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/carm1-in-6.html

• Smiles:

  CN(C)CCN(CC1)CCN1C2=NC=C(C(C3=CC=C(C)C=C3)=N2)C4=COC=C4

• Molecular Weight:

  391.51

• References & Citations:

  [1]Peng BL, et al. A CARM1 Inhibitor Potently Suppresses Breast Cancer Both In Vitro and In Vivo. J Med Chem. 2024 May 23;67(10):7921-7934.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported