Matriptase-IN-2 (free base)

• CAS Number:

  1268874-08-3

• UNSPSC Description:

  Matriptase-IN-2 free base is a matriptase inhibitor with a Ki of 5 nM. Matriptase-IN-2 has the potential for musculoskeletal system disorder research (WO2011023958A1; compound 432)[1].

• Target Antigen:

  Ser/Thr Protease

• Type:

  Reference compound

• Related Pathways:

  Metabolic Enzyme/Protease

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/matriptase-in-2-free-base.html

• Solubility:

  10 mM in DMSO

• Smiles:

  ClC1=C(C=CC(Cl)=C1)C2=CC=CC(S(N[C@H](C(N3CCC(CC3)CCN)=O)CC4=CC(C(N)=N)=CC=C4)(=O)=O)=C2

• Molecular Weight:

  602.58

• References & Citations:

  [1]Andrew David Rowan, et al. Screening methods. WO2011023958A1.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported